Carbolines. Part VII. Anisidines, convenient tools to synthesize hydroxy‐β‐carbolines

No Thumbnail Available
Date
1995-08
Authors
Rocca, P.
Marsais, F.
Godard, A.
Queguiner, G.
Adams, L.A.
Alo, B.I.
Journal Title
Journal ISSN
Volume Title
Publisher
Journal of Heterocyclic Chemistry
Abstract
The paper describes a convenient synthesis of hydroxy‐β‐carbolines from commercial anisidines based on key steps such as metalation, cross‐coupling and cyclization. The first total synthesis of a major cyto‐toxic constituent of a marine bryozoan is also reported, the 8‐hydroxy‐1‐vinyl‐β‐carboline.
Description
Keywords
Research Subject Categories::NATURAL SCIENCES::Chemistry::Organic chemistry , synthesis , anisidines , cyclization , cross‐coupling
Citation
Rocca, P., Marsais, F., Godard, A., Quéguiner, G., Adams, L., & Alo, B. (1995). Carbolines. Part VII. Anisidines, convenient tools to synthesize hydroxy‐β‐carbolines. Journal of heterocyclic chemistry, 32(4), 1171-1175.